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Protein kinase C inhibitors, their specificity and IC50 values. |
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| Inhibitor (Selectivity) |
IC50 Values |
Concentration Used |
Reference |
|
|
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| Gö6976 (α > β) |
PKCα = 2 nM; PKCβ1 = 6 nM |
3 nM |
[66, 67] |
| Hispidin (β) |
PKCβ = 3 μM |
6 μM |
[68] |
| Rottlerin (δ) |
PKCδ = 2–6μ M; PKCα,β,γ = 30–40 μM |
6 μM |
[51, 69] |
Mathison and Davison Journal of Inflammation 2006 3:9 doi:10.1186/1476-9255-3-9 |
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